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Variation in glucuronidation of lamotrigine in human liver microsomes
U. A. Argikar,
R. P. Remmel
Medicinal Chemistry
Carcinogenesis and Chemoprevention
Research output
:
Contribution to journal
›
Article
›
peer-review
60
Scopus citations
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Keyphrases
Lamotrigine
100%
Glucuronidation
100%
Human Liver Microsomes
100%
UGT1A4
50%
Antiepileptic Drugs
33%
Uridine
33%
Young Donors
33%
Formation Rate
33%
Elderly Donor
33%
Liquid Chromatography-tandem Mass Spectrometry (LC-MS/MS)
16%
Benzodiazepines
16%
Elderly Subjects
16%
Mass-based
16%
Glucuronide
16%
Therapeutic Concentrations
16%
Young Subjects
16%
Valproic Acid
16%
Triazine Ring
16%
Quaternary Ammonium Salt
16%
Liver Mass
16%
UGT1A3
16%
Intrinsic Clearance
16%
Lorazepam
16%
UGT2B7
16%
UGT2B4
16%
Diaminotriazine
16%
Pharmacology, Toxicology and Pharmaceutical Science
Lamictal
100%
Uridine
66%
Glucuronide
33%
Sodium Valproate
33%
Lorazepam
33%
Anticonvulsive Agent
33%
Intrinsic Clearance
33%
Quaternary Ammonium Derivative
33%
Triazine
33%