Translocation of ligand conformational free energy in receptor activation

A possible functional role of conformational isomerism in drug action

Research output: Contribution to journalArticle

7 Citations (Scopus)
Original languageEnglish (US)
Pages (from-to)806-807
Number of pages2
JournalJournal of Pharmaceutical Sciences
Volume60
Issue number5
DOIs
StatePublished - Jan 1 1971

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Isomerism
Drug Receptors
Energy Transfer
Structure-Activity Relationship
Theoretical Models
Pharmacology
Ligands
Pharmaceutical Preparations

Keywords

  • Conformation isomerism relationship—biological activity
  • Ligand conformational free energy—receptor activation

Cite this

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title = "Translocation of ligand conformational free energy in receptor activation: A possible functional role of conformational isomerism in drug action",
keywords = "Conformation isomerism relationship—biological activity, Ligand conformational free energy—receptor activation",
author = "Portoghese, {Philip S}",
year = "1971",
month = "1",
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language = "English (US)",
volume = "60",
pages = "806--807",
journal = "Journal of Pharmaceutical Sciences",
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publisher = "John Wiley and Sons Inc.",
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