Synthesis of Functionalized N-Arylsulfonyl Aziridines from α,β-Unsaturated Esters, Amides, Ketones, and Nitriles Using N,N-Dichloroarylsulfonamides as Nitrogen Source

Keyphrases

• Nitrogen Source 100%
• Ketones 100%
• Unsaturated Esters 100%
• Aziridine 100%
• Arylsulfonyl 100%
• α,β-unsaturated Amides 100%
• Unsaturated Nitriles 100%
• Olefins 50%
• Cyano 50%
• Cyclization 50%
• Good Yield 50%
• Acyl 50%
• Sodium Hydroxide 50%
• Stereoselectivity 50%
• Carboxamide 50%
• Alkoxycarbonyl 50%
• Aziridination 50%
• Sodium Sulfite 50%
• Cu(OAc)2 50%
• Sequence of Steps 50%

Chemistry

• Ketones 100%
• Carboxamide 100%
• Aziridine 100%
• Nitrile 100%
• Primary Structure 50%
• Alkene 50%