Solution-phase synthesis of chiral O-acyl isodipeptides

Mirna El Khatib, Lilibeth Jauregui, Srinivasa R. Tala, Levan Khelashvili, Alan R. Katritzky

Research output: Contribution to journalArticlepeer-review

22 Scopus citations

Abstract

O-Acylation of N-Boc-protected-serine and -threonine with N-Pg-(α-aminoacyl)benzotriazoles afforded the chiral O-acylated isodipeptides at 23 °C in yields of 74-91%.

Original languageEnglish (US)
Pages (from-to)1087-1092
Number of pages6
JournalMedChemComm
Volume2
Issue number11
DOIs
StatePublished - Nov 1 2011

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