N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442))

K. S. Thorneloe; A. C. Sulpizio; Z. Lin; D. J. Figueroa; A. K. Clouse; G. P. McCafferty; T. P. Chendrimada; E. S. Lashinger; E. Gordon; L. Evans; B. A. Misajet; D. J. DeMarini; J. H. Nation; L. N. Casillas; R. W. Marquis; B. J. Votta; S. A. Sheardown; X. Xu; D. P. Brooks; N. J. Laping; T. D. Westfall

N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442))

K. S. Thorneloe
, A. C. Sulpizio
, Z. Lin
, D. J. Figueroa
, A. K. Clouse
, G. P. McCafferty
, T. P. Chendrimada
, E. S. Lashinger
, E. Gordon
, L. Evans
, B. A. Misajet
, D. J. DeMarini
, J. H. Nation
, L. N. Casillas
, R. W. Marquis
, B. J. Votta
, S. A. Sheardown
, X. Xu
, D. P. Brooks
, N. J. Laping

T. D. Westfall

Research output: Contribution to journal › Comment/debate › peer-review

Original language	English (US)
Pages (from-to)	410
Number of pages	1
Journal	Journal of Pharmacology and Experimental Therapeutics
Volume	338
Issue number	1
State	Published - Jul 2011
Externally published	Yes

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Thorneloe, K. S., Sulpizio, A. C., Lin, Z., Figueroa, D. J., Clouse, A. K., McCafferty, G. P., Chendrimada, T. P., Lashinger, E. S., Gordon, E., Evans, L., Misajet, B. A., DeMarini, D. J., Nation, J. H., Casillas, L. N., Marquis, R. W., Votta, B. J., Sheardown, S. A., Xu, X., Brooks, D. P., ... Westfall, T. D. (2011). N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442)). Journal of Pharmacology and Experimental Therapeutics, 338(1), 410.

N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442)). / Thorneloe, K. S.; Sulpizio, A. C.; Lin, Z. et al.
In: Journal of Pharmacology and Experimental Therapeutics, Vol. 338, No. 1, 07.2011, p. 410.

Research output: Contribution to journal › Comment/debate › peer-review

Thorneloe, KS, Sulpizio, AC, Lin, Z, Figueroa, DJ, Clouse, AK, McCafferty, GP, Chendrimada, TP, Lashinger, ES, Gordon, E, Evans, L, Misajet, BA, DeMarini, DJ, Nation, JH, Casillas, LN, Marquis, RW, Votta, BJ, Sheardown, SA, Xu, X, Brooks, DP, Laping, NJ & Westfall, TD 2011, 'N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442))', Journal of Pharmacology and Experimental Therapeutics, vol. 338, no. 1, pp. 410.

Thorneloe KS, Sulpizio AC, Lin Z, Figueroa DJ, Clouse AK, McCafferty GP et al. N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442)). Journal of Pharmacology and Experimental Therapeutics. 2011 Jul;338(1):410.

Thorneloe, K. S. ; Sulpizio, A. C. ; Lin, Z. et al. / N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity : Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442)). In: Journal of Pharmacology and Experimental Therapeutics. 2011 ; Vol. 338, No. 1. pp. 410.

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title = "N-((1S)-1-\{[4-((2S)-2-\{[2,4-Dichlorophenyl)sulfonyl]amino\} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl\}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442))",

author = "Thorneloe, \{K. S.\} and Sulpizio, \{A. C.\} and Z. Lin and Figueroa, \{D. J.\} and Clouse, \{A. K.\} and McCafferty, \{G. P.\} and Chendrimada, \{T. P.\} and Lashinger, \{E. S.\} and E. Gordon and L. Evans and Misajet, \{B. A.\} and DeMarini, \{D. J.\} and Nation, \{J. H.\} and Casillas, \{L. N.\} and Marquis, \{R. W.\} and Votta, \{B. J.\} and Sheardown, \{S. A.\} and X. Xu and Brooks, \{D. P.\} and Laping, \{N. J.\} and Westfall, \{T. D.\}",

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month = jul,

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T1 - N-((1S)-1-{[4-((2S)-2-{[2,4-Dichlorophenyl)sulfonyl]amino} -3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl-1-benzothiophene-2- carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity

T2 - Part I (Journal of Pharmacology and Experimental Therapeutics (2008) 326, (432-442))

AU - Thorneloe, K. S.

AU - Sulpizio, A. C.

AU - Lin, Z.

AU - Figueroa, D. J.

AU - Clouse, A. K.

AU - McCafferty, G. P.

AU - Chendrimada, T. P.

AU - Lashinger, E. S.

AU - Gordon, E.

AU - Evans, L.

AU - Misajet, B. A.

AU - DeMarini, D. J.

AU - Nation, J. H.

AU - Casillas, L. N.

AU - Marquis, R. W.

AU - Votta, B. J.

AU - Sheardown, S. A.

AU - Xu, X.

AU - Brooks, D. P.

AU - Laping, N. J.

AU - Westfall, T. D.

PY - 2011/7

Y1 - 2011/7

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AN - SCOPUS:79959502564

SN - 0022-3565

VL - 338

SP - 410

JO - Journal of Pharmacology and Experimental Therapeutics

JF - Journal of Pharmacology and Experimental Therapeutics

IS - 1

ER -

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