Abstract
A systematic study of α-iodination and subsequent Suzuki-Miyaura couplings between non-attenuated enaminones and a wide range of aromatic boronic acids is reported. The microwave-assisted variant of this transformation furnished the α-arylenaminones in significantly shorter reaction times and slightly improved yields as compared to conventional heating.
Original language | English (US) |
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Pages (from-to) | 8811-8814 |
Number of pages | 4 |
Journal | Tetrahedron Letters |
Volume | 48 |
Issue number | 50 |
DOIs | |
State | Published - Dec 10 2007 |
Externally published | Yes |