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Discovery of Irreversible p97 Inhibitors
Rui Ding
, Ting Zhang
, Daniel J. Wilson
,
Jiashu Xie
,
Jessica Williams
, Yue Xu
, Yihong Ye
,
Liqiang Chen
Center for Drug Design
Carcinogenesis and Chemoprevention
Research output
:
Contribution to journal
›
Article
›
peer-review
20
Scopus citations
Overview
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Keyphrases
Amides
25%
Biological Evaluation
25%
Computer Modeling
25%
Covalent Inhibitor
25%
Cysteine Residues
25%
Design Evaluation
25%
In Cancer
25%
Irreversible Inhibitor
25%
Mass Spectrometry
25%
Mutagenesis
25%
New Inhibitors
25%
P97 Inhibitor
100%
Potential Therapeutics
25%
Reverse Amide
25%
Synthetic Evaluation
25%
Therapeutic Use
25%
Valosin-containing Protein
25%
Pharmacology, Toxicology and Pharmaceutical Science
Carboxamide
100%
Cysteine
50%
Diseases
50%
Malignant Neoplasm
50%
Mutagenesis
50%
Valosin Containing Protein
50%
Chemistry
Carboxamide
100%
Cysteine
50%
Mass Spectrometry
50%
Biochemistry, Genetics and Molecular Biology
Cysteine
14%
DNA Template
14%
Mass Spectrometry
14%
Mutagenesis
14%
P97
100%
Valosin-Containing Protein
14%