Aromatase inhibition by 4-thiosubstituted-4-androstene-3,17-dione derivatives

Keyphrases

• Inhibitory Activity 100%
• Androstenedione 100%
• 4-androstene-3,17-dione (4-AD) 100%
• Synthesized Compounds 100%
• Aromatase Inhibition 100%
• Estrogen 50%
• Synthetase 50%
• Competitive Inhibitor 50%
• Aromatase 50%
• Initial Velocity 50%
• 4-Androstenedione 50%
• Thiol Reagents 50%
• Microsomal Preparation 50%
• Enzyme Sources 50%
• Bulky Substituents 50%
• C-4 Position 50%

Pharmacology, Toxicology and Pharmaceutical Science

• Aromatase 100%
• Androstenedione 100%
• Competitive Inhibitor 20%
• Thiol Reagent 20%