Abstract
Attempted N,N-dibenzoylation of aminomethanesulfonic acid results in CS bond cleavage, generating synthetically useful α-benzamidomethylating electrophiles. The importance of this observation in regard to the reported failures to prepare sulfonamide analogs of peptides is discussed.
Original language | English (US) |
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Pages (from-to) | 537-540 |
Number of pages | 4 |
Journal | Tetrahedron Letters |
Volume | 22 |
Issue number | 6 |
DOIs | |
State | Published - 1981 |