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A 2-hydroxyisoquinoline-1,3-dione active-site RNase H inhibitor binds in multiple modes to HIV-1 reverse transcriptase

  • Karen A. Kirby
  • , Nataliya A. Myshakina
  • , Martin T. Christen
  • , Yue Lei Chen
  • , Hilary A. Schmidt
  • , Andrew D. Huber
  • , Zhaoyong Xi
  • , Seongmi Kim
  • , Rohit K. Rao
  • , Skyler T. Kramer
  • , Qiongying Yang
  • , Kamalendra Singh
  • , Michael A. Parniak
  • , Zhengqiang Wang
  • , Rieko Ishima
  • , Stefan G. Sarafianos

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Pharmacology, Toxicology and Pharmaceutical Science