1-Amido-3-(1H)-1,2-benziodoxoles: Stable amidoiodanes and reagents for direct amidation of organic substrates

Viktor Zhdankin, Marc McSherry, Brian Mismash, Jason T. Bolz, Jessica K. Woodward, Ruslan M. Arbit, Scott Erickson

Research output: Contribution to journalArticle

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Abstract

Amidobenziodoxoles 2 can be prepared from benziodoxole 1, trimethylsilyltriflate and the appropriate amides in the form of stable, microcrystalline compounds. Amidobenziodoxoles 2 react with adamantane 3 or N,N-dimethylarylamines 5 to afford the corresponding products of amidation, 4 and 6.

Original languageEnglish (US)
Pages (from-to)21-24
Number of pages4
JournalTetrahedron Letters
Volume38
Issue number1
DOIs
StatePublished - Jan 6 1997

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