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Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.

  • 4 Similar Profiles
Receptor, Serotonin, 5-HT2B Medicine & Life Sciences
Ursodeoxycholic Acid Medicine & Life Sciences
Protein-Serine-Threonine Kinases Medicine & Life Sciences
Prodrugs Medicine & Life Sciences
Bile Acids and Salts Medicine & Life Sciences
Testis Medicine & Life Sciences
Contraception Medicine & Life Sciences
Ligands Medicine & Life Sciences

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Research Output 2013 2017

18 Citations (Scopus)

BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen

Ayoub, A. M., Hawk, L. M. L., Herzig, R. J., Jiang, J., Wisniewski, A. J., Gee, C. T., Zhao, P., Zhu, J. Y., Berndt, N., Offei-Addo, N. K., Scott, T. G., Qi, J., Bradner, J. E., Ward, T. R., Schönbrunn, E., Georg, G. I. & Pomerantz, W. C. K., Jun 22 2017, In : Journal of Medicinal Chemistry. 60, 12, p. 4805-4817 13 p.

Research output: Contribution to journalArticle

Open Access
Ligands
Fluorescence Polarization
Uracil
Structure-Activity Relationship
Contraception
2 Citations (Scopus)

Potent Pyrimidine and Pyrrolopyrimidine Inhibitors of Testis-Specific Serine/Threonine Kinase 2 (TSSK2)

Hawkinson, J. E., Sinville, R., Mudaliar, D., Shetty, J., Ward, T., Herr, J. C. & Georg, G. I., Nov 22 2017, In : ChemMedChem. 12, 22, p. 1857-1865 9 p.

Research output: Contribution to journalArticle

Open Access
Protein-Serine-Threonine Kinases
Testis
Inhibitory Concentration 50
Staurosporine
Electrophoretic Mobility Shift Assay
15 Citations (Scopus)

Synthesis and Evaluation of Water-Soluble Prodrugs of Ursodeoxycholic Acid (UDCA), an Anti-apoptotic Bile Acid

Dosa, P. I., Ward, T., Castro, R. E., Rodrigues, C. M. P. & Steer, C. J., Jun 1 2013, In : ChemMedChem. 8, 6, p. 1002-1011 10 p.

Research output: Contribution to journalArticle

Ursodeoxycholic Acid
Prodrugs
Bile Acids and Salts
Water
Alkaline Phosphatase
14 Citations (Scopus)

Synthesis of novel analogs of cabergoline: Improving cardiovascular safety by removing 5-HT2B receptor agonism

Dosa, P. I., Ward, T., Walters, M. A. & Kim, S. W., Feb 14 2013, In : ACS Medicinal Chemistry Letters. 4, 2, p. 254-258 5 p.

Research output: Contribution to journalArticle

Receptor, Serotonin, 5-HT2B
Safety
Serotonin 5-HT2 Receptor Agonists
Prolactinoma
Pituitary ACTH Hypersecretion