19962020

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Article
2020

N-butyldeoxygalactonojirimycin induces reversible infertility in male CD rats

Gupta, V., Hild, S. A., Jakkaraj, S. R., Carlson, E. J., Wong, H. L., Allen, C. L., Georg, G. & Tash, J. S., Jan 1 2020, In : International Journal of Molecular Sciences. 21, 1, 301.

Research output: Contribution to journalArticle

Open Access
2018
Open Access
2 Scopus citations
2015

Scalable syntheses of the BET bromodomain inhibitor JQ1

Syeda, S. S., Jakkaraj, S. & Georg, G. I., May 25 2015, In : Tetrahedron Letters. 56, 23, p. 3454-3457 4 p.

Research output: Contribution to journalArticle

7 Scopus citations
2013

Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases

Schonbrunn, E., Betzi, S., Alam, R., Martin, M. P., Becker, A., Han, H., Francis, R., Chakrasali, R., Jakkaraj, S., Kazi, A., Sebti, S. M., Cubitt, C. L., Gebhard, A. W., Hazlehurst, L. A., Tash, J. S. & Georg, G. I., May 23 2013, In : Journal of medicinal chemistry. 56, 10, p. 3768-3782 15 p.

Research output: Contribution to journalArticle

39 Scopus citations
2011

Discovery of a potential allosteric ligand binding site in CDK2

Betzi, S., Alam, R., Martin, M., Lubbers, D. J., Han, H., Jakkaraj, S. R., Georg, G. I. & Schönbrunn, E., May 20 2011, In : ACS Chemical Biology. 6, 5, p. 492-501 10 p.

Research output: Contribution to journalArticle

95 Scopus citations
2008

A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose

Tash, J. S., Attardi, B., Hild, S. A., Chakrasali, R., Jakkaraj, S. R. & Georg, G., Jun 1 2008, In : Biology of Reproduction. 78, 6, p. 1127-1138 12 p.

Research output: Contribution to journalArticle

62 Scopus citations

Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat sertoli cells

Tash, J. S., Chakrasali, R., Jakkaraj, S. R., Hughes, J., Smith, S. K., Hornbaker, K., Heckert, L. L., Ozturk, S. B., Hadden, M. K., Kinzy, T. G., Blagg, B. S. J. & Georg, G., Jun 1 2008, In : Biology of Reproduction. 78, 6, p. 1139-1152 14 p.

Research output: Contribution to journalArticle

58 Scopus citations
1996
7 Scopus citations

Synthesis of 2-(3-aryl-4-formylpyrazol-1-yl)-3-phenyl-1,8-naphthyridines

Rao, J. S., Mogilaiah, K. & Sreenivasulu, B., Jul 1 1996, In : Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry. 35, 7, p. 713-714 2 p.

Research output: Contribution to journalArticle

6 Scopus citations