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Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.

  • 4 Similar Profiles
Histone Acetyltransferases Medicine & Life Sciences
4-Aminobenzoic Acid Medicine & Life Sciences
Peptides Chemical Compounds
Acetyl Coenzyme A Medicine & Life Sciences
Inhibitory Concentration 50 Medicine & Life Sciences
Molecular Imaging Medicine & Life Sciences
Triage Medicine & Life Sciences
High Fat Diet Medicine & Life Sciences

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Research Output 2006 2019

3,3′-Disubstituted 5,5′-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity

Xue, L., Shi, D. H., Harjani, J. R., Huang, F., Beveridge, J. G., Dingjan, T., Ban, K., Diab, S., Duffy, S., Lucantoni, L., Fletcher, S., Chiu, F. C. K., Blundell, S., Ellis, K., Ralph, S. A., Wirjanata, G., Teguh, S., Noviyanti, R., Chavchich, M., Creek, D. & 10 others, Price, R. N., Marfurt, J., Charman, S. A., Cuellar, M. E., Strasser, J. M., Dahlin, J. L., Walters, M. A., Edstein, M. D., Avery, V. M. & Baell, J. B., Jan 1 2019, In : Journal of Medicinal Chemistry.

Research output: Contribution to journalArticle

Antimalarials
Plasmodium falciparum
Plasmodium vivax
Triazines
Parasitemia

Discovery of benzoylsulfonohydrazides as potent inhibitors of the histone acetyltransferase KAT6A

Leaver, D. J., Cleary, B., Nguyen, N., Priebbenow, D. L., Lagiakos, H. R., Sanchez, J., Xue, L., Huang, F., Sun, Y., Mujumdar, P., Mudududdla, R., Varghese, S., Teguh, S., Charman, S. A., White, K. L., Katneni, K., Cuellar, M. E., Strasser, J. M., Dahlin, J. L., Walters, M. A. & 10 others, Street, I. P., Monahan, B. J., Jarman, K. E., Sabroux, H. J., Falk, H., Chung, M. C., Hermans, S. J., Parker, M. W., Thomas, T. & Baell, J. B., Aug 8 2019, In : Journal of Medicinal Chemistry. 62, 15, p. 7146-7159 14 p.

Research output: Contribution to journalArticle

Histone Acetyltransferases
Acetyl Coenzyme A
Inhibitory Concentration 50
Pharmaceutical Chemistry
Cell Aging

111 In-DANBIRT in Vivo Molecular Imaging of Inflammatory Cells in Atherosclerosis

Mota, R., Campen, M. J., Cuellar, M. E., Garver, W. S., Hesterman, J., Qutaish, M., Daniels, T., Nysus, M., Wagner, C. R. & Norenberg, J. P., Jan 1 2018, In : Contrast Media and Molecular Imaging. 2018, 6508724.

Research output: Contribution to journalArticle

Open Access
Molecular Imaging
High Fat Diet
Atherosclerotic Plaques
Atherosclerosis
Ozone
3 Citations (Scopus)

ALARM NMR for HTS triage and chemical probe validation

Dahlin, J. L., Cuellar, M. E., Singh, G., Nelson, K., Strasser, J. M., Rappe, T., Xia, Y., Veglia, G. & Walters, M. A., Mar 1 2018, In : Current protocols in chemical biology. 10, 1, p. 91-117 27 p.

Research output: Contribution to journalArticle

Open Access
Triage
Magnetic Resonance Spectroscopy
Proteins
Antigens
Sulfhydryl Compounds
25 Citations (Scopus)

Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors

Dahlin, J. L., Nelson, K. M., Strasser, J. M., Barsyte-Lovejoy, D., Szewczyk, M. M., Organ, S., Cuellar, M., Singh, G., Shrimp, J. H., Nguyen, N., Meier, J. L., Arrowsmith, C. H., Brown, P. J., Baell, J. B. & Walters, M. A., Dec 1 2017, In : Nature communications. 8, 1, 1527.

Research output: Contribution to journalArticle

Open Access
liabilities
Histone Acetyltransferases
inhibitors
Assays
counters