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Expertise related to UN Sustainable Development Goals
In 2015, UN member states agreed to 17 global Sustainable Development Goals (SDGs) to end poverty, protect the planet and ensure prosperity for all. This person’s work contributes towards the following SDG(s):
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The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.
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Collaborations and top research areas from the last five years
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Projects
- 1 Active
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Triptonide Prodrugs
Georg, G. (PI), Wong, H. L. (CoI), Jakkaraj, S. R. (Other Role), John, K. E. (Other Role) & Vantaddu, N. R. (Other Role)
12/15/24 → 5/31/25
Project: Research project
Research output
- 11 Article
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Incorporation of Three Extracyclic Arginine Residues into a Melanocortin Macrocyclic Agonist (c[Pro-His-DPhe-Arg-Trp-Dap-Lys(Arg-Arg-Arg-Ac)-DPro]) Decreases Food Intake When Administered Intrathecally or Subcutaneously Compared to a Macrocyclic Ligand Lacking Extracyclic Arginine Residues (c[Pro-His-DPhe-Arg-Trp-Dap-Ala-DPro)]
Ericson, M. D., Freeman, K. T., Larson, C. M., Bouchard, J. L., John, K., Lunzer, M. M., Koerperich, Z. M. & Haskell-Luevano, C., Apr 12 2024, In: ACS Pharmacology and Translational Science. 7, 4, p. 1114-1125 12 p.Research output: Contribution to journal › Article › peer-review
Open Access -
Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding
Faber, E. B., Sun, L., Tang, J., Roberts, E., Ganeshkumar, S., Wang, N., Rasmussen, D., Majumdar, A., Hirsch, L. E., John, K., Yang, A., Khalid, H., Hawkinson, J. E., Levinson, N. M., Chennathukuzhi, V., Harki, D. A., Schönbrunn, E. & Georg, G. I., Dec 2023, In: Nature communications. 14, 1, 3213.Research output: Contribution to journal › Article › peer-review
Open Access18 Scopus citations -
Discovery of a Pan-Melanocortin Receptor Antagonist [Ac-DPhe(pI)-Arg-Nal(2′)-Orn-NH2] at the MC1R, MC3R, MC4R, and MC5R that Mediates an Increased Feeding Response in Mice and a 40-Fold Selective MC1R Antagonist [Ac-DPhe(pI)-DArg-Nal(2′)-Arg-NH2]
Ericson, M. D., Tran, L. T., Mathre, S. S., Freeman, K. T., Holdaway, K., John, K., Lunzer, M. M., Bouchard, J. L. & Haskell-Luevano, C., Jun 22 2023, In: Journal of medicinal chemistry. 66, 12, p. 8103-8117 15 p.Research output: Contribution to journal › Article › peer-review
3 Scopus citations -
Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice
Faber, E. B., Wang, N., John, K., Sun, L., Wong, H. L., Burban, D., Francis, R., Tian, D., Hong, K. H., Yang, A., Wang, L., Elsaid, M., Khalid, H., Levinson, N. M., Schönbrunn, E., Hawkinson, J. E. & Georg, G. I., Feb 9 2023, In: Journal of medicinal chemistry. 66, 3, p. 1928-1940 13 p.Research output: Contribution to journal › Article › peer-review
15 Scopus citations -
Development of WEE2 kinase inhibitors as novel non-hormonal female contraceptives that target meiosis
Hanna, C. B., Mudaliar, D., John, K., Leigh Allen, C., Sun, L., Hawkinson, J. E., Schönbrunn, E., Georg, G. I. & Jensen, J. T., Aug 1 2020, In: Biology of reproduction. 103, 2, p. 368-377 10 p.Research output: Contribution to journal › Article › peer-review
Open Access10 Scopus citations