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Projects 2007 2021

Protein-Serine-Threonine Kinases
Contraception
Testis
Drug Discovery
Pharmaceutical Preparations
Male Contraceptive Agents
Cell Cycle
Phosphotransferases
Pharmaceutical Preparations

Research Output 1983 2018

Allosteric Modulators of Drug Targets Special Issue

Haskell-Luevano, C., Georg, G. I., Wang, S. & Meanwell, N. Feb 22 2018 In : Journal of Medicinal Chemistry. 61, 4, 1 p.

Research output: Contribution to journalEditorial

Pharmaceutical Preparations

Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception

Syeda, S. S., Sánchez, G., Hong, K. H., Hawkinson, J. E., Georg, G. I. & Blanco, G. Mar 8 2018 In : Journal of Medicinal Chemistry. 61, 5, p. 1800-1820 21 p.

Research output: Contribution to journalArticle

Ouabain
Contraception
Spermatozoa
Protein Isoforms
Sperm Tail

Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors

Chen, Y., Zhu, J. Y., Hong, K. H., Mikles, D. C., Georg, G. I., Goldstein, A. S., Amory, J. K. & Schönbrunn, E. Mar 16 2018 In : ACS chemical biology. 13, 3, p. 582-590 9 p.

Research output: Contribution to journalArticle

Slip forming
NAD
Tretinoin
Cracks
Catalytic Domain

Syntheses of PDE3A inhibitor ORG9935 and determination of the absolute stereochemistries of its enantiomers by X-ray crystallography

Jakkaraj, S. R., Young, V. G. & Georg, G. I. May 31 2018 In : Tetrahedron. 74, 22, p. 2769-2774 6 p.

Research output: Contribution to journalArticle

Slip forming
X Ray Crystallography
Chromatography
Pharmaceutical Preparations
thiophene-2-carboxylate
5 Citations

BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen

Ayoub, A. M., Hawk, L. M. L., Herzig, R. J., Jiang, J., Wisniewski, A. J., Gee, C. T., Zhao, P., Zhu, J. Y., Berndt, N., Offei-Addo, N. K., Scott, T. G., Qi, J., Bradner, J. E., Ward, T. R., Schönbrunn, E., Georg, G. I. & Pomerantz, W. C. K. Jun 22 2017 In : Journal of Medicinal Chemistry. 60, 12, p. 4805-4817 13 p.

Research output: Contribution to journalArticle

Ligands
Fluorescence Polarization
Uracil
Structure-Activity Relationship
Contraception