If you made any changes in Pure these will be visible here soon.

Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.

  • 4 Similar Profiles
Paclitaxel Medicine & Life Sciences
Microtubules Medicine & Life Sciences
Tubulin Medicine & Life Sciences
Cytotoxicity Chemical Compounds
beta-Lactams Chemical Compounds
Assays Chemical Compounds
docetaxel Medicine & Life Sciences
Taxoids Chemical Compounds

Network Recent external collaboration on country level. Dive into details by clicking on the dots.

Projects 2007 2021

Protein-Serine-Threonine Kinases
Drug Discovery
Pharmaceutical Preparations
Male Contraceptive Agents
Cell Cycle
Pharmaceutical Preparations

Research Output 1983 2018

Allosteric Modulators of Drug Targets Special Issue

Haskell-Luevano, C., Georg, G. I., Wang, S. & Meanwell, N. Feb 22 2018 In : Journal of Medicinal Chemistry. 61, 4, 1 p.

Research output: Contribution to journalEditorial

Pharmaceutical Preparations

Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception

Syeda, S. S., Sánchez, G., Hong, K. H., Hawkinson, J. E., Georg, G. I. & Blanco, G. Mar 8 2018 In : Journal of Medicinal Chemistry. 61, 5, p. 1800-1820 21 p.

Research output: Contribution to journalArticle

Protein Isoforms
Sperm Tail

Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors

Chen, Y., Zhu, J. Y., Hong, K. H., Mikles, D. C., Georg, G. I., Goldstein, A. S., Amory, J. K. & Schönbrunn, E. Mar 16 2018 In : ACS chemical biology. 13, 3, p. 582-590 9 p.

Research output: Contribution to journalArticle

Slip forming
Catalytic Domain

Syntheses of PDE3A inhibitor ORG9935 and determination of the absolute stereochemistries of its enantiomers by X-ray crystallography

Jakkaraj, S. R., Young, V. G. & Georg, G. I. May 31 2018 In : Tetrahedron. 74, 22, p. 2769-2774 6 p.

Research output: Contribution to journalArticle

Slip forming
X Ray Crystallography
Pharmaceutical Preparations
5 Citations

BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen

Ayoub, A. M., Hawk, L. M. L., Herzig, R. J., Jiang, J., Wisniewski, A. J., Gee, C. T., Zhao, P., Zhu, J. Y., Berndt, N., Offei-Addo, N. K., Scott, T. G., Qi, J., Bradner, J. E., Ward, T. R., Schönbrunn, E., Georg, G. I. & Pomerantz, W. C. K. Jun 22 2017 In : Journal of Medicinal Chemistry. 60, 12, p. 4805-4817 13 p.

Research output: Contribution to journalArticle

Fluorescence Polarization
Structure-Activity Relationship