1983 …2024
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Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.

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Projects 2007 2024

D3 Antagonist for Substance Use Disorder

Gurvich, V. J., Georg, G. & Walters, M. A.

NIH NIDA NATL INST ON DRUG AB

9/26/199/25/21

Project: Research project

Substance-Related Disorders

MASTER: CRO Support for NCATS Medicinal Chemistry for Lead Optimization

Gurvich, V. J., Georg, G., Hawkinson, J., Walters, M. A. & Wong, H. L.

NIHNIDA NATL INST ON DRUG AB

9/26/199/25/24

Project: Research project

Pharmaceutical Chemistry
Lead
National Center for Advancing Translational Sciences (U.S.)
Protein-Serine-Threonine Kinases
Contraception
Testis

Research Output 1983 2019

A Message from the Editors-in-Chief

Wang, S. & Georg, G., Mar 14 2019, In : Journal of Medicinal Chemistry. 62, 5, p. 2215-2216 2 p.

Research output: Contribution to journalEditorial

Drug Metabolism and Toxicology Special Issue Call for Papers

Guengerich, F. P., Georg, G. & Wang, S., Feb 14 2019, In : Journal of Medicinal Chemistry. 62, 3, 1 p.

Research output: Contribution to journalEditorial

Toxicology
Pharmaceutical Preparations
2 Citations (Scopus)

Identification of the Metabolic Profile of the α-Tubulin-Binding Natural Product (-)-Pironetin

Coulup, S. K., Huang, D. S., Wong, H. L. & Georg, G., Feb 14 2019, In : Journal of Medicinal Chemistry. 62, 3, p. 1684-1689 6 p.

Research output: Contribution to journalArticle

Metabolome
Tubulin
Biological Products
Liver Microsomes
Ovarian Neoplasms

Intranasal coadministration of a diazepam prodrug with a converting enzyme results in rapid absorption of diazepam in rats

Rautiola, D., Maglalang, P. D., Cheryala, N., Nelson, K. M., Georg, G. I., Fine, J. M., Svitak, A. L., Faltesek, K. A., Hanson, L. R., Mishra, U., Coles, L. D., Cloyd, J. C. & Siegel, R. A., Jan 1 2019, In : Journal of Pharmacology and Experimental Therapeutics. 370, 3, p. 796-805 10 p.

Research output: Contribution to journalArticle

Open Access
Prodrugs
Diazepam
Enzymes
Solubility
Pharmaceutical Preparations

Revisiting microtubule targeting agents: α-Tubulin and the pironetin binding site as unexplored targets for cancer therapeutics

Coulup, S. K. & Georg, G., Aug 1 2019, In : Bioorganic and Medicinal Chemistry Letters. 29, 15, p. 1865-1873 9 p.

Research output: Contribution to journalReview article

Tubulin
Microtubules
Binding Sites
Neoplasms
Therapeutics