1994 …2020
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Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.

Melanocortins Medicine & Life Sciences
Melanocortin Receptors Medicine & Life Sciences
Receptor, Melanocortin, Type 4 Medicine & Life Sciences
Agouti-Related Protein Medicine & Life Sciences
Melanocyte-Stimulating Hormones Medicine & Life Sciences
Ligands Medicine & Life Sciences
Peptides Medicine & Life Sciences
Receptor, Melanocortin, Type 3 Medicine & Life Sciences

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Projects 2011 2020

Melanocortin Receptors
Opioid Receptors
Pain
Therapeutics
Melanocortins
Defensins
Ligands
Melanocortins
Defensins
Ligands
Melanocortins
Ligands

Research Output 1994 2019

Allosteric Modulators of Drug Targets

Haskell-Luevano, C. & Meanwell, N. A., Oct 1 2019, In : Journal of Medicinal Chemistry. 62, 1, p. 1-2 2 p.

Research output: Contribution to journalEditorial

Pharmaceutical Preparations
1 Citation (Scopus)

Developing a Biased Unmatched Bivalent Ligand (BUmBL) Design Strategy to Target the GPCR Homodimer Allosteric Signaling (cAMP over β-Arrestin 2 Recruitment) Within the Melanocortin Receptors

Lensing, C. J., Freeman, K. T., Schnell, S. M., Speth, R. C., Zarth, A. T. & Haskell-Luevano, C., Jan 10 2019, In : Journal of Medicinal Chemistry. 62, 1, p. 144-158 15 p.

Research output: Contribution to journalArticle

Melanocortin Receptors
G-Protein-Coupled Receptors
Melanocortins
Ligands
Arrestin

Discovery of Polypharmacological Melanocortin-3 and -4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a μm MC4R Partial Agonist

Fleming, K. A., Freeman, K. T., Powers, M. D., Santos, R. G., Debevec, G., Giulianotti, M. A., Houghten, R. A., Doering, S. R., Pinilla, C. & Haskell-Luevano, C., Mar 14 2019, In : Journal of Medicinal Chemistry. 62, 5, p. 2738-2749 12 p.

Research output: Contribution to journalArticle

Receptor, Melanocortin, Type 3
Receptor, Melanocortin, Type 4
Melanocortins
Homeostasis
Molecular Probes
2 Citations (Scopus)

1,2,3-Triazole Rings as a Disulfide Bond Mimetic in Chimeric AGRP-Melanocortin Peptides: Design, Synthesis, and Functional Characterization

Tala, S. R., Singh, A., Lensing, C. J., Schnell, S. M., Freeman, K. T., Rocca, J. R. & Haskell-Luevano, C., May 16 2018, In : ACS Chemical Neuroscience. 9, 5, p. 1001-1013 13 p.

Research output: Contribution to journalArticle

Melanocortins
Triazoles
Melanocortin Receptors
Disulfides
Peptides

Allosteric Modulators of Drug Targets Special Issue

Haskell-Luevano, C., Georg, G. I., Wang, S. & Meanwell, N., Feb 22 2018, In : Journal of Medicinal Chemistry. 61, 4, 1 p.

Research output: Contribution to journalEditorial

Pharmaceutical Preparations