Projects per year
Fingerprint The Fingerprint is created by mining the titles and abstracts of the person's research outputs and projects/funding awards to create an index of weighted terms from discipline-specific thesauri.
Melanocortins
Medicine & Life Sciences
Melanocortin Receptors
Medicine & Life Sciences
Receptor, Melanocortin, Type 4
Medicine & Life Sciences
Agouti-Related Protein
Medicine & Life Sciences
Ligands
Medicine & Life Sciences
Melanocyte-Stimulating Hormones
Medicine & Life Sciences
Peptides
Medicine & Life Sciences
Receptor, Melanocortin, Type 3
Medicine & Life Sciences
Network
Recent external collaboration on country level. Dive into details by clicking on the dots.
Projects 2011 2020
Novel Melanocortin Receptor Probe Discovery
NIH Natl Inst of Diabetes/Dig/Kidney Dis
4/1/16 → 3/31/20
Project: Research project
Melanocortin Receptors
Discovery of Opioid Receptor Endogenous Allosteric Modul
Winston & Maxine Wallin Neuro Disc Fund
1/1/18 → 12/31/18
Project: Research project
Opioid Receptors
Pain
Therapeutics
Defensins as Melanocortin Ligands
NIH Natl Inst of Diabetes/Dig/Kidney Dis
10/1/15 → 11/30/17
Project: Research project
Melanocortins
Defensins
Ligands
Defensins as Melanocortin Ligands
NIH Natl Inst of Diabetes/Dig/Kidney Dis
12/1/12 → 11/30/15
Project: Research project
Melanocortins
Defensins
Ligands
Melanocortin Selective Ligands
NIH Natl Inst of Diabetes/Dig/Kidney Dis
5/1/12 → 4/30/17
Project: Research project
Melanocortins
Ligands
Research Output 1994 2019
Allosteric Modulators of Drug Targets
Haskell-Luevano, C. & Meanwell, N. A., Oct 1 2019, In : Journal of Medicinal Chemistry. 62, 1, p. 1-2 2 p.Research output: Contribution to journal › Editorial
Pharmaceutical Preparations
1
Citation
(Scopus)
Developing a Biased Unmatched Bivalent Ligand (BUmBL) Design Strategy to Target the GPCR Homodimer Allosteric Signaling (cAMP over β-Arrestin 2 Recruitment) Within the Melanocortin Receptors
Lensing, C. J., Freeman, K. T., Schnell, S. M., Speth, R. C., Zarth, A. T. & Haskell-Luevano, C., Jan 10 2019, In : Journal of Medicinal Chemistry. 62, 1, p. 144-158 15 p.Research output: Contribution to journal › Article
Melanocortin Receptors
G-Protein-Coupled Receptors
Melanocortins
Ligands
Arrestin
1
Citation
(Scopus)
Discovery of Polypharmacological Melanocortin-3 and -4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a μm MC4R Partial Agonist
Fleming, K. A., Freeman, K. T., Powers, M. D., Santos, R. G., Debevec, G., Giulianotti, M. A., Houghten, R. A., Doering, S. R., Pinilla, C. & Haskell-Luevano, C., Mar 14 2019, In : Journal of Medicinal Chemistry. 62, 5, p. 2738-2749 12 p.Research output: Contribution to journal › Article
Receptor, Melanocortin, Type 3
Receptor, Melanocortin, Type 4
Melanocortins
Homeostasis
Molecular Probes
Structure–activity relationships of the tetrapeptide Ac-His-Arg-(Pi)Dphe-TiC-NH 2 at the mouse melanocortin receptors: Modification at the (PI)DPhe position leads to MMC3R versus MMC4R selective ligands
Schlasner, K. N., Ericson, M. D., Doering, S. R., Freeman, K. T., Weinrich, M. & Haskell-Luevano, C., Apr 13 2019, In : Molecules. 1463.Research output: Contribution to journal › Article
Open Access
Melanocortin Receptors
mice
food intake
knockout mice
Ligands
2
Citations
(Scopus)
1,2,3-Triazole Rings as a Disulfide Bond Mimetic in Chimeric AGRP-Melanocortin Peptides: Design, Synthesis, and Functional Characterization
Tala, S., Singh, A., Lensing, C. J., Schnell, S. M., Freeman, K. T., Rocca, J. R. & Haskell-Luevano, C., May 16 2018, In : ACS Chemical Neuroscience. 9, 5, p. 1001-1013 13 p.Research output: Contribution to journal › Article
Melanocortins
Triazoles
Melanocortin Receptors
Disulfides
Peptides