Projects per year
- 50 - 100 out of 284 results
Search results
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Finished
Discovery and development of allosteric inhibitors of Cdk2/cyclin E as non-toxic ovarian cancer drugs
Georg, G. (PI), Hawkinson, J. (CoI) & Wong, H. L. (CoI)
7/1/22 → 6/30/23
Project: Research project
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Midwest AViDD Center
Harris, R. (PI), Aihara, H. (CoI), Aliota, M. T. (CoI), Harki, D. A. (CoI), Langlois, R. A. (CoI), Li, F. (CoI), Liang, Y. (CoI) & Ly, H. (CoI)
NIH Nat'l Inst of Allergy & Infect Dis
5/16/22 → 4/30/25
Project: Research project
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Biochar as a tool for preventing root infection of soybean seedlings by Macrophomina phaseolina andother soil fungi
Shier, T. (PI)
USDA AGRICULTURAL RESEARCH SERVICE, MISSISSIPPI SOYBEAN PROMOTION BOARD
10/1/21 → 1/31/22
Project: Research project
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Development/Validation of Rete Testis Microcannulation for the Assessment of Novel Chemical Scaffolds That Penetrate the Blood Testis Barrier
Wong, H. L. (PI) & Georg, G. (CoI)
NIH NAT'L INST OF CHILD HEALTH/HUMAN DEV
9/17/21 → 9/16/23
Project: Research project
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Development of Probes to Characterize the Role of HINT1 in Mu Opioid Receptor and N-Methyl-D-Aspartate Receptor Cross-Regulation
Dillenburg, M. D. (PI)
AMERICAN FDN FOR PHARMACEUTICAL EDUC
9/1/21 → 8/31/22
Project: Research project
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Predictive Models for Small-Molecule Accumulation in Gram-Negative Bacteria
Duerfeldt, A. S. (PI)
MEMORIAL SLOAN-KETTERING CANCER CENTER, NATIONAL INSTITUTES OF HEALTH (NIH)
8/1/21 → 7/31/24
Project: Research project
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Identification of novel dual-acting bactericidal drug targets for tuberculosis treatment
Baughn, A. (PI) & Aldrich, C. (CoI)
FUJITA HEALTH UNIVERSITY, GLOBAL HEALTH INNOVATIVE TECHNOLOGY FUND
7/6/21 → 1/31/25
Project: Research project
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Melanocortin Receptor Selective Ligands
Haskell-Luevano, C. (PI)
NATIONAL INSTITUTES OF HEALTH (NIH)
7/1/21 → 4/30/25
Project: Research project
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Harnessing N-Myc Signaling by Chemical Degradation of Aurora Kinase A
Harki, D. A. (PI)
AMERICAN ASSOCIATION FOR CANCER RESEARCH
7/1/21 → 6/30/22
Project: Research project
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A novel TNFR1-selective small molecule inhibitor to treat rheumatoid arthritis and related inflammatory diseases
Binstadt, B. A. (PI), Sachs, J. N. (CoI) & Ferguson, D. M. (Other Role)
RHEUMATOLOGY RESEARCH FOUNDATION
7/1/21 → 6/30/24
Project: Research project
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Mycotoxin production by the soybean red leaf blotch fungus Coniothyrium glycines
Shier, T. (PI)
USDA AGRICULTURAL RESEARCH SERVICE
4/7/21 → 4/30/24
Project: Research project
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Small Molecule PPAR-alpha Agonism as a Novel Approach to Treat Eye Vascular Diseases
Duerfeldt, A. S. (PI)
3/1/21 → 4/30/25
Project: Research project
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Chemical probes as allosteric modulators of CK2 alpha prime targeting Huntington's disease
Walters, M. A. (PI), Finzel, B. C. (CoI) & Nelson, K. (Prior Principal Investigator)
NIH NAT INST OF NEURO DISORDERS & STROKE
2/15/21 → 1/31/23
Project: Research project
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Drug Discovery Pipeline Targeting Pathologically Leaky Calcium Release Channels in Age-Related Indications
Aldrich, C. (PI)
PHOTONIC PHARMA LLC, NATIONAL INSTITUTES OF HEALTH (NIH)
1/15/21 → 12/31/22
Project: Research project
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Development of New Alpha 4 Inhibitor Compound and Selectivity Assay for Male Contraception
Georg, G. (PI), Hawkinson, J. (CoI) & Wong, H. L. (CoI)
1/5/21 → 7/1/22
Project: Research project
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Rifamycins for NTM and PROTACS for mycobacteria
Aldrich, C. (PI)
HACKENSACK MERIDIAN HEALTH, INC
1/1/21 → 12/31/22
Project: Research project
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A Novel Small Molecule for The Prevention and Treatment of Diabetic Retinopathy
Duerfeldt, A. S. (PI)
EXCITANT THERAPEUTICS LLC, NATIONAL INSTITUTES OF HEALTH (NIH)
1/1/21 → 2/28/22
Project: Research project
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A Novel Small Molecule for The Prevention and Treatment of Age-Related Macular Degeneration
Duerfeldt, A. S. (PI)
EXCITANT THERAPEUTICS LLC, NATIONAL INSTITUTES OF HEALTH (NIH)
1/1/21 → 8/31/22
Project: Research project
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Evaluating therapeutic potential of a novel PPAR-a agonist for wet-AMD
Duerfeldt, A. S. (PI)
EXCITANT THERAPEUTICS LLC, NATIONAL INSTITUTES OF HEALTH (NIH)
1/1/21 → 2/28/22
Project: Research project
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The Role of HIF1A-DNMT3A axis in AML1/ETO-Driven Acute Myelogenous Leukemia
Liu, S. (PI), Tretyakova, N. Y. (CoI) & Yang, R. (CoI)
NIH NATIONAL CANCER INSTITUTE (NCI)
12/7/20 → 8/28/22
Project: Research project
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Chemical Methods to Characterize Penicillin-Binding Protein Function and Interactions
Carlson, E. E. (PI) & Ambrose, E. A. (CoI)
NIH NIGMS NATL INST OF GENERAL
9/18/20 → 6/30/24
Project: Research project
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Development of Methods for the Efficient Capture and Analysis of Circulating Breast Cancer Tumor Cells
Wagner, C. R. (PI)
MAYO CLINIC ROCHESTER, NIH NATIONAL CANCER INSTITUTE (NCI)
9/1/20 → 8/31/21
Project: Research project
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Targeting Na,K-ATPase alpha4 for male contraception
Georg, G. (PI) & Wong, H. L. (CoI)
UNIVERSITY OF KANSAS MEDICAL CENTER, NATIONAL INSTITUTES OF HEALTH (NIH)
8/15/20 → 4/30/25
Project: Research project
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Structural Dynamics of Muscle Calcium ATPase Regulation
Thomas, D. D. (PI), Aihara, H. (CoI), Cornea, R. L. (Co-Principal Investigator) & Aldrich, C. (Consultant/Collaborator)
NIH NAT'L HEART, LUNG, AND BLOOD INSTITU
5/1/20 → 4/30/24
Project: Research project
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Identification of mycotoxins used in soybean root infection by Macrophomina phaseolina and other fungi
Shier, T. (PI)
MISSISSIPPI STATE UNIVERSITY, MISSISSIPPI SOYBEAN PROMOTION BOARD
4/1/20 → 3/31/21
Project: Research project
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Membrane-active quinoline and quinazoline antibacterials that target Gram positive pathogens
Aldrich, C. (PI)
DARTMOUTH COLLEGE, NATIONAL INSTITUTES OF HEALTH (NIH)
3/1/20 → 2/28/25
Project: Research project
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Time-resolved FRET-based allostery sensors for any protein kinase drug target
Levinson, N. M. (PI), Drake, J. M. (CoI), Georg, G. (CoI) & Thomas, D. D. (CoI)
NIH NATIONAL CANCER INSTITUTE (NCI)
3/1/20 → 2/29/24
Project: Research project
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Functions of CD177 as a novel IgG Fc receptor
Wu, J. (PI) & Hawkinson, J. (CoI)
NIH Nat'l Inst of Allergy & Infect Dis
2/21/20 → 1/31/23
Project: Research project
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Overcoming Pyrazinamide Resistance with Pyrazinoate-Cephalosporin Conjugates
Aldrich, C. (PI), Baughn, A. (CoI) & Ferguson, D. M. (CoI)
NIH Nat'l Inst of Allergy & Infect Dis
1/25/20 → 12/31/21
Project: Research project
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Optimization of the Composition of Corn Starch-based Bioplastic to ControlAflatoxin and Other Agricultural Pests
Shier, T. (PI)
USDA AGRICULTURAL RESEARCH SERVICE
10/1/19 → 6/30/21
Project: Research project
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Mechanisms of PhIP-induced dopaminergic neurotoxicity
Turesky, R. (PI)
PURDUE UNIVERSITY, NATIONAL INSTITUTES OF HEALTH (NIH)
10/1/19 → 5/31/22
Project: Research project
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MASTER: CRO Support for NCATS Medicinal Chemistry for Lead Optimization
Gurvich, V. J. (PI), Georg, G. (CoI), Hawkinson, J. (CoI), Walters, M. A. (CoI) & Wong, H. L. (CoI)
9/26/19 → 4/28/25
Project: Research project
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D3 Antagonist for Substance Use Disorder
Gurvich, V. J. (PI), Georg, G. (CoI) & Walters, M. A. (CoI)
9/26/19 → 9/25/21
Project: Research project
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Allosteric CDK2 inhibitor Discovery and Development for Male Contraception
Georg, G. (PI) & Wong, H. L. (CoI)
NIH NAT'L INST OF CHILD HEALTH/HUMAN DEV
9/13/19 → 8/31/21
Project: Research project
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Minnesota HHEAR Targeted Analysis Laboratory
Peterson, L. A. (PI), Balbo, S. (CoI), Gross, M. D. (CoI), Hecht, S. S. (CoI), Murphy, S. E. (CoI), Stepanov, I. (CoI), Turesky, R. (CoI) & Villalta, P. W. (CoI)
NIH NATL INST OF ENVIRON HEALTH SCIENCES
9/5/19 → 3/31/25
Project: Research project
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Profiling DNA adducts in formalin fixed paraffin embedded human colorectal tissue
Turesky, R. (PI) & Yun, B. (CoI)
NIH NATIONAL CANCER INSTITUTE (NCI)
9/1/19 → 8/31/22
Project: Research project
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APOBEC MUTAGENESIS IN BREAST CANCER
Harris, R. (PI), Aihara, H. (CoI), Harki, D. A. (CoI), Largaespada, D. A. (CoI) & Yee, D. (CoI)
NIH NATIONAL CANCER INSTITUTE (NCI)
8/9/19 → 7/31/22
Project: Research project
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NF-kappaB Inducing Kinase (NIK) for the Treatment of Hematologic Malignancies
Tang, J. (PI)
7/1/19 → 6/30/21
Project: Research project
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Chemical Inhibition of APOBEC-catalyzed Tumor Evolution
Harki, D. A. (PI)
AMERICAN ASSOCIATION FOR CANCER RESEARCH
7/1/19 → 6/30/20
Project: Research project
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Development of Allosteric Inhibitors against Cyclin-Dependent Kinase 2 (Cdk2)
Faber, E. (PI)
NIH NATIONAL CANCER INSTITUTE (NCI)
7/1/19 → 6/30/22
Project: Research project
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Target based discovery of next generation pyrazinamide
Aldrich, C. (PI)
HACKENSACK MERIDIAN HEALTH, INC, NATIONAL INSTITUTES OF HEALTH (NIH)
6/1/19 → 5/31/23
Project: Research project
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DNA adductome of human bladder from the tobacco exposome
Turesky, R. (PI), Bellamri, M. (CoI) & Yun, B. (CoI)
NIH NATL INST OF ENVIRON HEALTH SCIENCES
4/1/19 → 12/31/24
Project: Research project
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Identification of mycotoxins used in soybean root infection by Macrophomina phaseolina and other fungi
Shier, T. (PI)
MISSISSIPPI STATE UNIVERSITY, MISSISSIPPI SOYBEAN PROMOTION BOARD
4/1/19 → 6/30/20
Project: Research project
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Homogeneous Screening Assay for Cytokine Receptor Modulators
Hawkinson, J. (PI)
STATEGICS, INC, NATIONAL INSTITUTES OF HEALTH (NIH)
3/1/19 → 2/28/22
Project: Research project
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Caspase-2 Probe Compounds
Ashe, K. H. (PI), Finzel, B. C. (CoI) & Nelson, K. (CoI)
NIH NAT'L INSTITUTE ON AGING (NIA)
2/15/19 → 11/30/24
Project: Research project
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Chromatin regions, genes and pathways that confer susceptibility to chemical-induced DNA damage
Tretyakova, N. Y. (PI)
TEXAS A & M UNIVERSITY, NATIONAL INSTITUTES OF HEALTH (NIH)
2/1/19 → 1/31/25
Project: Research project
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Cancer Center Support Grant
Yee, D. (PI), AbuSalah, A. M. (CoI), Basu, S. (CoI), Beckman, K. B. (CoI), Bielinsky, A. K. (CoI), Cooley, S. A. (CoI), De For, T. E. (CoI), Falconer, S. N. (CoI), Felices, M. (CoI), Griffin, T. J. (CoI), Hallstrom, T. C. (CoI), Hatsukami, D. K. (CoI), Hendrickson, E. A. (CoI), Hirsch, B. A. (CoI), Joseph, A. M. (CoI), Kirstein, M. N. (CoI), Konety, B. R. (CoI), Koopmeiners, J. (CoI), Kuntz, K. M. (CoI), Lange, C. A. (CoI), Largaespada, D. A. (CoI), Le, C. T. (CoI), LeBeau, A. (CoI), Lindgren, B. R. (CoI), Luo, X. (CoI), Mc Carthy, J. B. (CoI), McKenna, D. H. (CoI), Miller, J. S. (CoI), Moriarity, B. S. (CoI), Nelson, H. H. (CoI), O'Sullivan, G. (CoI), Ondrey, F. G. (CoI), Pennell, C. A. (CoI), Petersen, A. J. (CoI), Peterson, L. A. (CoI), Peterson, B. A. (CoI), Sarver, A. L. (CoI), Shimizu, Y. (CoI), Siegfried, J. M. (CoI), Temiz, N. A. (CoI), Turesky, R. (CoI), Vogel, R. (CoI), Wagner, J. E. (CoI), Wang, J. (CoI), Weigel, B. J. (CoI), Weisdorf, D. J. (CoI), Woo, J. (CoI) & Yamamoto, M. (CoI)
NIH NATIONAL CANCER INSTITUTE (NCI)
2/1/19 → 1/31/24
Project: Research project
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Gut Microbiota and Effect on Immune Suppressants in Transplantation
Jacobson, P. A. (PI), Matas, A. J. (CoI) & Remmel, R. P. (CoI)
HENNEPIN HEALTHCARE RESEARCH INSTITUTE, NATIONAL INSTITUTES OF HEALTH (NIH)
2/1/19 → 8/31/24
Project: Research project